SCHEMBL6174674

SCHEMBL6174674

CCc1ccc2[nH]c(C(=O)c3cc(C)ccn3)c(C(C)C(=O)O)c2c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.68
PTGS1 P23219 7/20 0.68
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
UTS2R Q9UKP6 1/20 0.35
TLR8 Q9NR97 2/20 0.35
TLR7 Q9NYK1 2/20 0.35
EGFR P00533 1/20 0.35
CDK2 P24941 1/20 0.35
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171474 0.93 PTGS2 (0.58) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL6171712 0.92 PTGS2 (0.68) PTGS2PTGS1AKR1C3AKR1C2
SCHEMBL6170712 0.89 PTGS2 (0.53) PTGS2PTGS1KDM4EALDH1A1NPC1
SCHEMBL6172560 0.85 PTGS2 (0.50) PTGS2PTGS1KDM4EGAATLR8
SCHEMBL6169271 0.85 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL6171752 0.85 PTGS2 (0.49) PTGS2PTGS1KDM4EALDH1A1MAPT
SCHEMBL6171838 0.84 PTGS2 (0.67) PTGS2PTGS1TLR8TLR7
SCHEMBL7202770 0.84 PTGS2 (0.48) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL6168891 0.84 PTGS2 (0.67) PTGS2PTGS1AKR1C2KDM4EALDH1A1
SCHEMBL6171485 0.83 PTGS2 (0.56) PTGS2PTGS1TLR8TLR7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed