SCHEMBL6169536

SCHEMBL6169536

CCCCCNc1nc(CC)c(-c2cc3c(cc2O)CCCC3)nc1CC

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 6/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
ACHE P22303 7/20 0.34
TLR7 Q9NYK1 1/20 0.33
BCHE P06276 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166393 0.87 CRHR1 (0.42) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6165792 0.86 KDM4E (0.40) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6167259 0.84 CRHR1 (0.44) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6165056 0.84 CRHR1 (0.43) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6169750 0.83 KDM4E (0.40) KDM4EALDH1A1HPGDACHEBCHE
SCHEMBL6168821 0.81 KDM4E (0.36) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6165798 0.79 CRHR1 (0.61) CRHR1
SCHEMBL6167908 0.77 CRHR1 (0.34) CRHR1KDM4EALDH1A1HPGD
SCHEMBL6166528 0.75 CRHR1 (0.43) CRHR1KDM4EALDH1A1HPGDACHE
SCHEMBL6168389 0.73 KDM4E (0.41) CRHR1KDM4EALDH1A1HPGDACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499599-A1 SUBSTITUTED PYRAZINE DERIVATIVES Pharmacia & Upjohn Company LLC (US) 2005-01-26 EP claimed
WO-2003091225-A1 SUBSTITUTED PYRAZINE DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 2003-11-06 WO claimed
EP-1499599-A1 SUBSTITUTED PYRAZINE DERIVATIVES Pharmacia & Upjohn Company LLC (US) 2005-01-26 EP disclosed
WO-2003091225-A1 SUBSTITUTED PYRAZINE DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 2003-11-06 WO disclosed