SCHEMBL6169705

SCHEMBL6169705

O=CNC1=CCC(c2ccccc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.38
SRD5A1 P18405 2/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.35
SLC18A3 Q16572 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C1 Q04828 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTRB1 P17538 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
HPGD P15428 1/20 0.32
SRD5A2 P31213 1/20 0.32
ADRA1A P35348 2/20 0.32
DAPK3 O43293 1/20 0.32
JAK2 O60674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10041970 0.75 NAPRT (0.41) SRD5A1KDM4ESLC18A3LMNAMAPT
SCHEMBL9518144 0.75 TRPA1 (0.44) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1
SCHEMBL7975812 0.71 SRD5A1 (0.37) SRD5A1KDM4ESLC18A3SIGMAR1GAA
SCHEMBL6740701 0.68 SLC18A3 (0.41) GRIN2BSRD5A1SLC18A3SIGMAR1LMNA
SCHEMBL9876026 0.68 SRD5A1 (0.43) GRIN2BSRD5A1ALDH1A1SLC18A3SIGMAR1
SCHEMBL24105190 0.68 SLC18A3 (0.41) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1
SCHEMBL17440328 0.68 SLC18A3 (0.41) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1
SCHEMBL17440329 0.68 SLC18A3 (0.41) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1
SCHEMBL25073357 0.68 SLC18A3 (0.41) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1
SCHEMBL9372709 0.68 GAA (0.41) GRIN2BSRD5A1KDM4ESLC18A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6914160-B1 Oxytocin inhibitors PFIZER INC (US) 2005-07-05 US disclosed
EP-1537085-A1 OXYTOCIN INHIBITORS Pfizer Limited (GB) 2005-06-08 EP disclosed
WO-2004020414-A1 OXYTOCIN INHIBITORS PFIZER LIMITED (GB) 2004-03-11 WO disclosed
WO-2000002864-A1 PRECUSORS FOR PNA-MONOMERS MARTENS JUERGEN (DE) 2000-01-20 WO disclosed