SCHEMBL6170101

SCHEMBL6170101

COc1ccc(-c2noc(SCc3ccsc3)c2-c2ccc(S(N)(=O)=O)cc2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.50
PTGS1 P23219 13/20 0.50
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
CDK2 P24941 1/20 0.40
ABCB11 O95342 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8474199 0.87 PTGS2 (0.42) PTGS2PTGS1CA12CA1CA2
SCHEMBL6170654 0.82 PTGS2 (0.55) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL8474198 0.81 PTGS2 (0.41) PTGS2PTGS1CA1
SCHEMBL6170119 0.80 PTGS2 (0.53) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6170018 0.78 PTGS2 (0.52) PTGS2PTGS1CDK2
SCHEMBL4888565 0.77 PTGS2 (0.67) PTGS2PTGS1CA12CA1CA2
SCHEMBL6169938 0.77 PTGS2 (0.58) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6168801 0.77 PTGS2 (0.55) PTGS2PTGS1CDK2
SCHEMBL6168516 0.77 PTGS2 (0.55) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6171523 0.76 PTGS2 (0.54) PTGS2PTGS1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1528059-A2 Substituted isoxazoles for the treatment of inflammation G.D. Searle LLC (US) 2005-05-04 EP disclosed
EP-1223167-A2 Substituted isoxazoles for the treatment of inflammation G.D. Searle & Co. (US) 2002-07-17 EP disclosed
US-5985902-A TREATING INFLAMMATION AND INFLAMMATION-ASSOCIATED DISORDERS, SUCH AS ARTHRITIS G.D. SEARLE & CO. (US) 1999-11-16 US disclosed