SCHEMBL61714

SCHEMBL61714

[O-][S+](Cc1ccc(O)cc1)Cc1ccc(O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.50
ESR2 Q92731 2/20 0.50
ABAT P80404 1/20 0.46
CA2 P00918 4/20 0.44
TAAR1 Q96RJ0 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
IDO1 P14902 2/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
SLC6A2 P23975 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR3A P46098 1/20 0.42
BACE1 P56817 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
BLM P54132 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
CA12 O43570 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11360108 0.81 CA2 (0.50) ESR1ESR2ABATCA2BLM
SCHEMBL777796 0.74 IDO1 (0.46) TAAR1IDO1LMNA
SCHEMBL4401171 0.74 IDO1 (0.46) CA2TAAR1ALDH1A1IDO1KMT2A
Benzene SCHEMBL11030926 0.72 CALM1 (0.45) TAAR1ALDH1A1IDO1SLC6A2HPGD
SCHEMBL22250999 0.72 ESR1 (0.54) ESR1ESR2CA2TAAR1KDM4E
SCHEMBL3387953 0.69 IDO1 (0.52) CA2TAAR1KDM4EALDH1A1IDO1
Ethane SCHEMBL7199050 0.68 TP53 (0.43) TAAR1KDM4EALDH1A1IDO1SLC6A2
SCHEMBL3873458 0.67 ESR1 (1.00) ESR1ESR2ABATCA2TAAR1
SCHEMBL69344 0.67 ESR1 (1.00) ESR1ESR2ABATCA2TAAR1
SCHEMBL2969737 0.67 ESR1 (1.00) ESR1ESR2ABATCA2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112190570-B Application of gastrodia tuber source derivative in preparing medicine for treating acute or chronic pain 中国医学科学院药物研究所 2023-05-05 CN disclosed
CN-112190570-A Application of derivative derived from rhizoma gastrodiae in preparation of medicine for treating acute or chronic pain 中国医学科学院药物研究所 2021-01-08 CN disclosed
CN-103420805-A Polybenzyl derivatives with nerve cell protective activity in tall gastrodia tuber INST MATERIA MEDICA CAMS 2013-12-04 CN disclosed
US-8129357-B2 N6-(4-hydroxybenzyl)adenosine; Gastrodia extract; neurodegenerative Huntington's disease; trinucleotide repeat disease; hypoglycemic; neurological antiinflammatory; amination of 6-chloropurine ribonucleoside with 4-hydroxybenzylamine; condensation of adenosine with 4-methoxybenzoyl chloride ACADEMIA SINICA (TW) 2012-03-06 US disclosed
US-20080176816-A1 Method of making and using an adenosine analogue ACADEMIA SINICA 2008-07-24 US disclosed
US-7351434-B2 Therapeutic Gastrodia extracts ACADEMIA SINICA (TW) 2008-04-01 US disclosed
US-20070237840-A1 Administering bis(4-hydroxybenzyl)sulfide for therapy of Huntington's disease ACADEMIA SINICA (TW) 2007-10-11 US disclosed
US-6242654-B1 REACTING A PHENOLATE COMPOUND WITH AN ORGANIC FLUORINATING AGENT TO PREPARE A FLUORINE SUBSTITUTED AROMATIC COMPOUND MITSUI CHEMICALS, INC. (JP) 2001-06-05 US disclosed
EP-1013629-A1 Preparation process of fluorine subsituted aromatic compound Mitsui Chemicals, Inc. (JP) 2000-06-28 EP disclosed
US-4302448-A Secretin preparations with intensified and protracted action, process for their manufacture, their use as well as dihydroxybenzoyl-L-tyrosine HOECHST AKTIENGESELLSCHAFT (DE) 1981-11-24 US disclosed
EP-0021184-A1 Pharmaceutical compositions based on secretin with enhanced and protracted activity, process for their preparation and dihydroxybenzoyl-L-tyrosine HOECHST AKTIENGESELLSCHAFT (DE) 1981-01-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176816-A1 Method of making and using an adenosine analogue HTT, ADA, GDA ESR1 4462/4885ESR2 3928/4885ABAT 145/4885
US-20070237840-A1 Administering bis(4-hydroxybenzyl)sulfide for therapy of Huntington's disease HTT, SNCA, SLC2A4 ESR1 3557/4885ESR2 2970/4885ABAT 42/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.