SCHEMBL6172162

SCHEMBL6172162

CC(=O)On1nnc(-c2ccccn2)n1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 11/20 0.47
HDAC6 Q9UBN7 2/20 0.45
TP53 P04637 1/20 0.43
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3585013 0.75 TP53 (0.55) GRM5TP53
SCHEMBL29972774 0.75 TP53 (0.55) GRM5TP53
SCHEMBL4699461 0.73 GRM5 (0.73) GRM5
SCHEMBL9542013 0.72 TSHR (0.46) TP53ALDH1A1
SCHEMBL6669232 0.72 GRM5 (0.69) GRM5
SCHEMBL6175160 0.72 MGLL (0.49) ALDH1A1
SCHEMBL5579857 0.70 HDAC6 (0.58) GRM5HDAC6ALDH1A1
SCHEMBL3585009 0.68 TP53 (0.55) GRM5TP53ALDH1A1
SCHEMBL14350435 0.68 HDAC6 (0.53) GRM5HDAC6TP53
SCHEMBL27916227 0.68 KDM4E (0.50) TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534693-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2005-06-01 EP claimed
WO-2004022523-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2004-03-18 WO claimed