SCHEMBL6173377

SCHEMBL6173377

CC(c1ccncc1NS(=O)(=O)N1CCOCC1)C1(C(C)c2ccncc2NS(=O)(=O)N2CCOCC2)NC(=O)N(c2ccc(OC(F)(F)F)cc2)C1=O

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 4/20 0.34
PKM P14618 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CCR9 P51686 2/20 0.33
CYP11B2 P19099 1/20 0.33
AKT1 P31749 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
ABL1 P00519 1/20 0.31
POLB P06746 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6172850 0.88 IGF1R (0.35) CYP2C9CYP2C19CYP11B2
SCHEMBL6174307 0.85 CYP2C9 (0.38) LIPEALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL6169571 0.84 CYP3A4 (0.35) LIPEALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL6173842 0.83 PRKDC (0.36) ALDH1A1CYP2C9CYP2C19CYP3A4GAA
SCHEMBL6173283 0.82 CYP3A4 (0.38) LIPEALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL6175672 0.81 LIPE (0.34) LIPEPKMCYP2C9CYP2C19CCR9
SCHEMBL6175670 0.81 MMP12 (0.34) LIPEPKMALDH1A1CYP2C9CYP2C19
SCHEMBL6178460 0.81 LIPE (0.38) LIPEALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL6173454 0.80 CYP2C9 (0.41) LIPEALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL6172844 0.79 CYP3A4 (0.40) ALDH1A1CYP2C9CYP2C19CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed