SCHEMBL6174587

SCHEMBL6174587

CC(c1ccncc1-c1ccc(Cl)cc1)C1(C(C)c2ccncc2-c2ccc(Cl)cc2)NC(=O)N(c2ccc(OC(F)(F)F)cc2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.37
GAA P10253 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPBWR1 P48145 1/20 0.35
MCHR1 Q99705 1/20 0.35
MARS1 P56192 1/20 0.34
CHRNA7 P36544 1/20 0.34
ENPP2 Q13822 1/20 0.34
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
CTSD P07339 3/20 0.33
BACE1 P56817 3/20 0.33
BACE2 Q9Y5Z0 3/20 0.33
LMNA P02545 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174506 0.92 CYP3A4 (0.43) MAPTGAACYP3A4CYP2C9CYP2C19
SCHEMBL6171727 0.92 HSD11B1 (0.36) GAACYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6174812 0.91 ALDH1A1 (0.38) GAACYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6172582 0.87 ALDH1A1 (0.36) GAACYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6174915 0.85 MAPT (0.38) MAPTGAACYP3A4CYP2C9CYP2C19
SCHEMBL6173429 0.84 POLB (0.41) MAPTGAACYP3A4CYP2C9CYP2C19
SCHEMBL6173440 0.83 CYP3A4 (0.38) GAACYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6175217 0.82 GAA (0.42) MAPTGAACYP3A4CYP2C9CYP2C19
SCHEMBL6173690 0.82 CYP3A4 (0.41) MAPTGAACYP3A4CYP2C9CYP2C19
SCHEMBL2941010 0.81 CYP3A4 (0.36) GAACYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed