SCHEMBL6175263

SCHEMBL6175263

CC(=O)Oc1ccc2oc(-c3ccc(F)cc3)nc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.55
TP53 P04637 6/20 0.55
CETP P11597 1/20 0.53
UTRN P46939 4/20 0.52
HTR2B P41595 1/20 0.52
HSD17B10 Q99714 3/20 0.52
THRB P10828 3/20 0.52
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 3/20 0.52
HPGD P15428 2/20 0.52
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
HDAC6 Q9UBN7 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
TSHR P16473 1/20 0.49
RXFP1 Q9HBX9 2/20 0.48
POLB P06746 1/20 0.48
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4032178 0.82 MAPT (0.60) MAPTTP53UTRNHTR2BHSD17B10
SCHEMBL27652488 0.82 HSD17B10 (0.70) MAPTTP53CETPUTRNHTR2B
SCHEMBL9112906 0.81 HSD17B10 (0.54) MAPTTP53CETPUTRNHTR2B
SCHEMBL9001602 0.80 MAPT (0.53) MAPTTP53CETPHSD17B10THRB
SCHEMBL9514445 0.79 MAPT (0.65) MAPTTP53HSD17B10KDM4EALDH1A1
SCHEMBL13254495 0.77 KDM4E (0.59) MAPTTP53UTRNHTR2BHSD17B10
SCHEMBL5638115 0.77 MAPT (0.70) MAPTTP53UTRNHTR2BHSD17B10
SCHEMBL18309416 0.76 MAPT (0.50) MAPTTP53CETPUTRNHTR2B
SCHEMBL12608957 0.76 MAOA (0.67) MAPTTP53UTRNHTR2BHSD17B10
SCHEMBL1675515 0.76 MAPT (0.65) MAPTTP53HSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1732161-A 1,3-diamino-2-hydroxypropane pro-drug derivatives ELAN PHARM INC (US) 2006-02-08 CN claimed
EP-1534693-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2005-06-01 EP claimed
WO-2004022523-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2004-03-18 WO claimed
CN-1732161-A 1,3-diamino-2-hydroxypropane pro-drug derivatives ELAN PHARM INC (US) 2006-02-08 CN disclosed