SCHEMBL6176299

SCHEMBL6176299

Cc1oc(=O)cc(O)c1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
GLA P06280 1/20 0.43
PIM1 P11309 1/20 0.43
ALDH1A1 P00352 8/20 0.41
KDM4E B2RXH2 8/20 0.41
HPGD P15428 4/20 0.41
MCL1 Q07820 4/20 0.41
HSD17B10 Q99714 3/20 0.41
THRB P10828 1/20 0.41
AKR1B1 P15121 1/20 0.41
GAA P10253 6/20 0.40
MAPT P10636 3/20 0.40
MAPK1 P28482 3/20 0.40
HTT P42858 3/20 0.40
LMNA P02545 2/20 0.40
NSD2 O96028 1/20 0.40
POLB P06746 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574998 0.77 CYP3A4 (0.46) CYP3A4KMT2AMEN1GLAALDH1A1
SCHEMBL9788316 0.71 ALDH1A1 (0.56) CYP3A4KMT2AMEN1ALDH1A1KDM4E
SCHEMBL7963459 0.71 ALDH1A1 (0.45) CYP3A4KMT2AMEN1GLAALDH1A1
SCHEMBL7968690 0.71 MEN1 (0.48) CYP3A4KMT2AMEN1GLAALDH1A1
SCHEMBL1804389 0.65
SCHEMBL24376358 0.63 CYP3A4 (0.45) CYP3A4KMT2AMEN1GLAALDH1A1
SCHEMBL2761996 0.63 ALDH1A1 (0.61) CYP3A4KMT2AMEN1GLAPIM1
SCHEMBL25581857 0.63 ACHE (0.43) CYP3A4KMT2AMEN1ALDH1A1KDM4E
SCHEMBL28794852 0.63 SELL (0.58) CYP3A4KMT2AMEN1PIM1ALDH1A1
SCHEMBL13824371 0.62 KDM4E (0.46) CYP3A4KMT2AMEN1GLAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1205198-C Cyclic ketone derivative and pharmaceutical use thereof TORAY INDUSTRIES (JP) 2005-06-08 CN disclosed
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP disclosed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP disclosed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
US-6184245-B1 Cyclic ketone derivatives and their medical applications TORAY INDUSTRIES INC. (JP) 2001-02-06 US disclosed
CN-1242770-A Cyclic ketone derivative and pharmaceutical use thereof TORAY INDUSTRIES (JP) 2000-01-26 CN disclosed
EP-0962456-A1 CYCLIC KETONE DERIVATIVE AND PHARMACEUTICAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 1999-12-08 EP disclosed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed