SCHEMBL6177670

SCHEMBL6177670

CC(=O)Nc1c(-c2ccncc2)c(-c2ccc(F)c(Cl)c2)nn1C.c1cc2cc-2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.43
ABL1 P00519 1/20 0.43
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
MAPK14 Q16539 4/20 0.39
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP17A1 P05093 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
BRAF P15056 2/20 0.37
CNR1 P21554 1/20 0.36
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180521 0.91 MAPK14 (0.41) ABL1ADORA3ADORA2AADORA2BADORA1
SCHEMBL4343334 0.87 MAPK14 (0.52) ADORA3ADORA2AADORA2BADORA1MAPK14
SCHEMBL6179168 0.82 NR3C1 (0.40) ABL1MAPK14MEN1MAPTKMT2A
SCHEMBL6179160 0.82 MAPK14 (0.46) MAPK14MAPT
SCHEMBL6177661 0.82 MAPK14 (0.57) MAPK14
SCHEMBL6173798 0.81 MAPK14 (0.42) ABL1MAPK14MEN1MAPTKMT2A
SCHEMBL6176926 0.81 MAPK14 (0.43) MAPK14MEN1MAPTKMT2ALMNA
SCHEMBL6173808 0.79 MAPT (0.36) ABL1MAPK14MEN1MAPTKMT2A
SCHEMBL6176923 0.79 P2RX7 (0.45) MAPK14
SCHEMBL7139557 0.78 MAPK14 (0.52) ADORA3ADORA2AADORA2BADORA1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142890-B1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG CO LTD (JP) 2005-08-03 EP disclosed
US-6511997-B1 For treatment of a disease associated with tumor necrosis factor alpha, interleukin 1, interleukin 6 or cyclooxygenase II; such as irritable bowel disease TEIKOKU HORMONE MFG. CO., LTD. (JP) 2003-01-28 US disclosed
EP-1142890-A1 AMINOPYRAZOLE DERIVATIVES TEIKOKU HORMONE MFG. CO., LTD. (JP) 2001-10-10 EP disclosed