SCHEMBL6177904

SCHEMBL6177904

CCOC(=O)C(=CNC1CC1)C(=O)c1cc(Br)c(F)c(Cl)c1F.CCOC(=O)c1cn(C2CC2)c2c(Cl)c(F)c(Br)cc2c1=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.45
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
KMT2A Q03164 2/20 0.34
TOP2A P11388 4/20 0.33
TOP2B Q02880 4/20 0.33
STAT3 P40763 1/20 0.33
KCNH2 Q12809 1/20 0.33
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4476600 0.85 ADRB2 (0.55) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL6475919 0.83 GPR35 (0.37) ALDH1A1POLBKMT2ALMNA
SCHEMBL4464475 0.83 GPR35 (0.37) ALDH1A1POLBKMT2ALMNA
SCHEMBL6166978 0.80 ADRB2 (0.49) ADRB2ALDH1A1POLBOPRM1KMT2A
SCHEMBL7575069 0.76 ADRB2 (0.61) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL10472998 0.76 ADRB2 (0.57) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL4564641 0.76 ADRB2 (0.57) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL7584091 0.74 ADRB2 (0.57) ADRB2ALDH1A1POLBCHRM2CHRM1
SCHEMBL8437121 0.74 POLB (0.39) ALDH1A1POLBKMT2ALMNA
SCHEMBL8436286 0.74 MAPT (0.36) ALDH1A1POLBKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532137-A2 ANTIMICROBIAL AZA-BICYCLIC DERIVATES, THEIR COMPOSITIONS AND USES THE PROCTER & GAMBLE COMPANY (US) 2005-05-25 EP disclosed
WO-2004014893-A2 ANTIMICROBIAL AZA-BICYCLIC DERIVATES, THEIR COMPOSITIONS AND USES THE PROCTER & GAMBLE COMPANY (US) 2004-02-19 WO disclosed