SCHEMBL6178375

SCHEMBL6178375

O=CCc1ccccc1Nc1nc(Cl)ncc1[N+](=O)[O-]

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 13/20 0.60
GSK3B P49841 1/20 0.43
IGF1R P08069 1/20 0.41
PRKCQ Q04759 3/20 0.40
MAPK1 P28482 2/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2916138 0.83 ALK (0.39) PIN1MAPT
SCHEMBL6176285 0.81 IGF1R (0.48) PIN1IGF1R
SCHEMBL18181774 0.76 PIN1 (0.63) PIN1GSK3BIGF1RMAPK1MAPT
SCHEMBL3811561 0.76 PIN1 (0.67) PIN1GSK3BIGF1RMAPK1MAPT
SCHEMBL3976795 0.76 PIN1 (1.00) PIN1GSK3BMAPK1MAPTL3MBTL1
SCHEMBL3814860 0.75 PIN1 (0.62) PIN1GSK3BIGF1RMAPK1MAPT
SCHEMBL1037559 0.75 PIN1 (0.65) PIN1GSK3BL3MBTL1
SCHEMBL1204172 0.75 PIN1 (0.62) PIN1GSK3BIGF1RMAPK1
Hydrochloric Acid SCHEMBL6178818 0.75 PTK2 (0.67) GSK3BIGF1RPRKCQMAPK1
SCHEMBL21846996 0.74 PIN1 (0.59) PIN1MAPK1MAPTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597251-A2 PYRIMIDINE COMPOUNDS SmithKline Beecham Corporation (US) 2005-11-23 EP disclosed
WO-2004074244-A2 PYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-09-02 WO disclosed