SCHEMBL6179979

SCHEMBL6179979

CC(C)(C)C(=O)CN1C(=O)C(N)CN(C(=O)C(C)(C)C)c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
CCKAR P32238 7/20 0.36
CCKBR P32239 6/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
THRB P10828 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177709 0.86 CCKBR (0.43) CCKBRPOLB
SCHEMBL6178279 0.84 CYP3A4 (0.37) ALDH1A1CCKBRMEN1KMT2A
SCHEMBL6176423 0.82 ALDH1A1 (0.48) ALDH1A1CCKARCCKBRTHRBPOLB
SCHEMBL1394353 0.82 ALDH1A1 (0.48) ALDH1A1CCKARCCKBRTHRBPOLB
SCHEMBL6175102 0.80 TSHR (0.43) ALDH1A1
SCHEMBL6180323 0.80 ALDH1A1 (0.46) ALDH1A1CCKARCCKBRMEN1KMT2A
SCHEMBL6180501 0.80 CCKBR (0.44) ALDH1A1CCKARCCKBRPOLB
Hydrochloric Acid SCHEMBL4423682 0.80 EGFR (0.41) CCKBRMEN1KMT2A
Hydrochloric Acid SCHEMBL4423689 0.80 EGFR (0.41) CCKBRMEN1KMT2A
SCHEMBL541718 0.79 CCKBR (0.46) ALDH1A1CCKARCCKBRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945445-B9 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2005-12-28 EP disclosed
EP-0945445-B1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARM CO LTD (JP) 2003-09-03 EP disclosed
US-6239131-B1 WHICH HAVE GASTRIN AND/OR CCK-B (CHOLECYSTOKININ-B) RECEPTOR ANTAGONISM, USEFUL AS REMEDIES FOR GASTRIC ULCER AND GASTROINTESTINAL MOVEMENT DISORDER. ZERIA PHARMACEUTICAL CO., LTD. (JP) 2001-05-29 US disclosed
EP-0945445-A1 1,5-BENZODIAZEPINE DERIVATIVES ZERIA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed