SCHEMBL6180217

SCHEMBL6180217

CC(C)(C)N(C(=O)O)[C@H](Cc1ccc(Cl)c(Cl)c1)C(=O)N1CCC[C@H]1C(=O)NCC1CCc2n[nH]cc2C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.38
SCN3A Q9NY46 1/20 0.38
TACR1 P25103 5/20 0.38
ALDH1A1 P00352 1/20 0.36
F2 P00734 7/20 0.35
XIAP P98170 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
BDKRB2 P30411 1/20 0.34
BDKRB1 P46663 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
F10 P00742 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
BUB1 O43683 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178779 0.90 TACR1 (0.38) TACR1ALDH1A1F2XIAPTAAR1
SCHEMBL6181640 0.85 F2 (0.39) SCN5ASCN3AF2
SCHEMBL6093180 0.85 TAAR1 (0.41) SCN5ASCN3ATACR1F2XIAP
Hydrochloric Acid SCHEMBL6093286 0.85 DPP4 (0.40) SCN5ASCN3AF2
SCHEMBL6179624 0.81 F2 (0.41) SCN5ASCN3AF2SMN1; SMN2PRSS1
SCHEMBL6181452 0.80 XIAP (0.40) TACR1F2XIAPPRSS1
SCHEMBL6180898 0.76 SCN4A (0.38) TACR1XIAPTAAR1
SCHEMBL6179716 0.75 DPP4 (0.41) XIAP
SCHEMBL6093203 0.75 XIAP (0.43) TACR1XIAPTAAR1
SCHEMBL6178208 0.75 XIAP (0.43) TACR1XIAPTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1287018-B1 THROMBIN INHIBITORS LEK TOVARNA FARMACEVTSKIH (SI) 2005-01-19 EP claimed