SCHEMBL6178779

SCHEMBL6178779

CC(C)(C)N(C(=O)O)[C@H](Cc1ccc(Cl)c(Cl)c1)C(=O)N1CCC[C@H]1C(=O)NC1CCc2n[nH]cc2C1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.38
SCN4A P35499 1/20 0.36
XIAP P98170 2/20 0.36
ALDH1A1 P00352 1/20 0.34
CASP1 P29466 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TAAR1 Q96RJ0 2/20 0.32
HTT P42858 1/20 0.32
UTS2R Q9UKP6 1/20 0.32
F2 P00734 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181452 0.90 XIAP (0.40) TACR1SCN4AXIAPF2
SCHEMBL6180217 0.90 SCN5A (0.38) TACR1XIAPALDH1A1TAAR1F2
SCHEMBL6180898 0.86 SCN4A (0.38) TACR1SCN4AXIAPCASP1TAAR1
SCHEMBL6179716 0.85 DPP4 (0.41) SCN4AXIAPHTT
SCHEMBL6093203 0.85 XIAP (0.43) TACR1XIAPTAAR1
SCHEMBL6178208 0.85 XIAP (0.43) TACR1XIAPTAAR1
Hydrochloric Acid SCHEMBL6196562 0.85 DPP4 (0.42) SCN4AXIAPHTT
Hydrochloric Acid SCHEMBL6094296 0.85 DPP4 (0.42) SCN4AXIAPHTT
SCHEMBL6178104 0.79 SCN4A (0.39) SCN4AXIAPCYP1A2CYP3A4CYP2D6
SCHEMBL6180622 0.79 SCN4A (0.39) SCN4AXIAPCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1287018-B1 THROMBIN INHIBITORS LEK TOVARNA FARMACEVTSKIH (SI) 2005-01-19 EP claimed