SCHEMBL6180506

SCHEMBL6180506

CCN(CC)CCCOC1(c2ccc3ccccc3c2)C(=O)N(C)c2cc(Cl)cc(Cl)c21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 3/20 0.45
SRC P12931 10/20 0.39
FGFR1 P11362 9/20 0.39
KDM4E B2RXH2 1/20 0.35
CCR2 P41597 4/20 0.34
EGFR P00533 2/20 0.34
FGFR2 P21802 2/20 0.34
FGFR4 P22455 2/20 0.34
FGFR3 P22607 2/20 0.34
MEN1 O00255 1/20 0.34
PIM1 P11309 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CHEK1 O14757 1/20 0.33
RIPK2 O43353 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180394 0.81 FGFR1 (0.39) GHSRSRCFGFR1KDM4ECCR2
SCHEMBL6180949 0.74 GHSR (0.54) GHSRMEN1KMT2A
SCHEMBL6177738 0.72 GHSR (0.45) GHSRKMT2A
SCHEMBL6178245 0.66 GHSR (0.58) GHSRMEN1PIM1KMT2ATDP1
SCHEMBL6176281 0.65 GHSR (0.43) GHSR
SCHEMBL6180015 0.64 GHSR (0.53) GHSRKMT2A
SCHEMBL6180568 0.64 GHSR (0.61) GHSRMEN1KMT2A
SCHEMBL6177474 0.64 GHSR (0.61) GHSRMEN1KMT2A
SCHEMBL6179661 0.64 GHSR (0.65) GHSRMEN1KMT2A
SCHEMBL6181396 0.63 GHSR (0.54) GHSRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-B1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMA (JP) 2005-02-09 EP disclosed
US-6576656-B1 Such as 1-(2-diethylaminoethyl)-4-trifluoromethyl-6-carbamoyl-3-hydroxy-3-(2 -chlorophenyl)oxindole; growth hormone releaser SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2003-06-10 US disclosed