SCHEMBL6180394

SCHEMBL6180394

CCN(CC)CCCOC1(c2ccc3ccccc3c2)C(=O)Nc2cc(Cl)cc(Cl)c21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.39
SRC P12931 3/20 0.39
GHSR Q92847 4/20 0.38
HTR6 P50406 6/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
HTR1A P08908 1/20 0.35
DRD1 P21728 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
CCR2 P41597 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180506 0.81 GHSR (0.45) FGFR1SRCGHSRKDM4ECCR2
SCHEMBL6176281 0.79 GHSR (0.43) GHSRMAOAMAOB
SCHEMBL6180564 0.70 ALDH1A1 (0.46) GHSRHTR6ALDH1A1TP53MAPT
SCHEMBL6180949 0.68 GHSR (0.54) GHSRHTR1A
SCHEMBL6180123 0.68 GHSR (0.69) GHSR
SCHEMBL30186208 0.63 KDM4E (0.62) KDM4EALDH1A1MAPTMAOB
SCHEMBL7855737 0.61 GHSR (0.78) GHSR
SCHEMBL21171901 0.59 SCN1A (0.46) KDM4EALDH1A1MAOBHTR1AHTR2A
SCHEMBL3973547 0.57 POLB (0.49) GHSRTP53MAPT
SCHEMBL29625659 0.57 KDM4E (0.60) KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-B1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMA (JP) 2005-02-09 EP disclosed
US-6576656-B1 Such as 1-(2-diethylaminoethyl)-4-trifluoromethyl-6-carbamoyl-3-hydroxy-3-(2 -chlorophenyl)oxindole; growth hormone releaser SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2003-06-10 US disclosed
EP-1105376-A1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-06-13 EP disclosed
WO-2000010975-A1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2000-03-02 WO disclosed