SCHEMBL6180591

SCHEMBL6180591

Cc1cccc(C2CCCN2S(=O)(=O)c2ccc(C)c(O)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
PSEN1 P49768 1/20 0.46
PSEN2 P49810 1/20 0.46
APH1B Q8WW43 1/20 0.46
NCSTN Q92542 1/20 0.46
APH1A Q96BI3 1/20 0.46
PSENEN Q9NZ42 1/20 0.46
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
HTR7 P34969 1/20 0.43
DRD3 P35462 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43
LOXL2 Q9Y4K0 2/20 0.42
NR3C2 P08235 1/20 0.42
HCRTR1 O43613 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178979 0.90 PSEN1 (0.57) TRPA1LMNAPSEN1PSEN2APH1B
SCHEMBL6179184 0.87 TRPA1 (0.57) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6178957 0.86 TRPA1 (0.56) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6178952 0.86 TRPA1 (0.56) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6178012 0.84 CYP3A4 (0.62) TRPA1LMNAMAPTKDM4ETP53
SCHEMBL6176638 0.82 TRPA1 (0.70) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6179258 0.82 PSEN1 (0.67) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6176643 0.82 TRPA1 (0.70) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6179250 0.82 PSEN1 (0.67) TRPA1LMNAMAPTPSEN1PSEN2
SCHEMBL6180434 0.81 TRPA1 (0.47) TRPA1LMNAPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165510-B1 1-ARENESULFONYL-2-ARYL-PYRROLIDINE AND PIPERIDINE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS HOFFMANN LA ROCHE (CH) 2005-09-28 EP claimed