SCHEMBL6178979

SCHEMBL6178979

Cc1ccc(S(=O)(=O)N2CCCC2c2ccccc2)cc1O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.57
PSEN2 P49810 1/20 0.57
APH1B Q8WW43 1/20 0.57
NCSTN Q92542 1/20 0.57
APH1A Q96BI3 1/20 0.57
PSENEN Q9NZ42 1/20 0.57
TRPA1 O75762 3/20 0.54
ACLY P53396 1/20 0.50
LOXL2 Q9Y4K0 2/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
NR3C2 P08235 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.43
USP2 O75604 1/20 0.43
ADRB2 P07550 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179184 0.90 TRPA1 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6180591 0.90 TRPA1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6178012 0.87 CYP3A4 (0.62) TRPA1CYP3A4CYP2C19LMNAALDH1A1
SCHEMBL6178185 0.86 TRPA1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6180434 0.84 TRPA1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6177618 0.82 PSEN1 (0.69) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6177624 0.82 PSEN1 (0.69) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6180512 0.81 LMNA (0.65) TRPA1LMNAALDH1A1GAAPOLB
SCHEMBL3370579 0.80 MAPT (0.48) NPSR1ALDH1A1GAAPOLB
SCHEMBL6180588 0.80 PSEN1 (0.74) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165510-B1 1-ARENESULFONYL-2-ARYL-PYRROLIDINE AND PIPERIDINE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS HOFFMANN LA ROCHE (CH) 2005-09-28 EP claimed