SCHEMBL6181682

SCHEMBL6181682

Cc1ccc(C(=O)c2sc(Nc3ccc(O[C@@H](C)C4CCCN4)cc3)nc2N)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
NPC1 O15118 3/20 0.51
TUBB8B A6NNZ2 1/20 0.50
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBB6 Q9BUF5 1/20 0.50
TUBB2B Q9BVA1 1/20 0.50
TUBB1 Q9H4B7 1/20 0.50
SPHK2 Q9NRA0 1/20 0.50
SPHK1 Q9NYA1 1/20 0.50
CDK5 Q00535 6/20 0.46
CDK5R1 Q15078 6/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181680 1.00 MEN1 (0.51) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6181787 0.88 CCNA2 (0.59) MEN1KMT2ANPC1CDK5CDK5R1
SCHEMBL6181795 0.88 CCNA2 (0.59) MEN1KMT2ANPC1CDK5CDK5R1
SCHEMBL6179405 0.87 CDK5 (0.51) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6179401 0.87 CDK5 (0.51) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6181893 0.84 CDK5 (0.50) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6182925 0.84 CDK5 (0.50) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6181454 0.84 ZAP70 (0.53) MEN1KMT2ANPC1TUBB8BTUBB4A
SCHEMBL6181449 0.84 ZAP70 (0.53) MEN1KMT2ANPC1TUBB8BTUBB4A
Acetic Acid SCHEMBL6179980 0.82 TUBB8B (0.46) MEN1KMT2ANPC1TUBB8BTUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507530-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-02-23 EP claimed
WO-2003097048-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-27 WO claimed
EP-1507530-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-02-23 EP disclosed
WO-2003097048-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-27 WO disclosed