SCHEMBL6183995

SCHEMBL6183995

COc1cnc(O)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.41
HPGD P15428 3/20 0.39
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
ALDH1A1 P00352 2/20 0.36
PTPN1 P18031 2/20 0.36
ALOX5 P09917 2/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
PDK2 Q15119 1/20 0.35
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
NNMT P40261 1/20 0.34
F2 P00734 1/20 0.34
GLA P06280 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5164798 0.78 CA12 (0.41) CYP3A4HPGDNOS3NOS1NOS2
SCHEMBL7940187 0.77 ALDH1A1 (0.39) CYP3A4NOS3NOS1NOS2ALDH1A1
SCHEMBL18679972 0.76 LMNA (0.34) ALDH1A1KMT2A
SCHEMBL7321441 0.76 MAPT (0.39) CYP3A4ALDH1A1CCR1CCR5CCR8
SCHEMBL23948543 0.74 NOS3 (0.56) NOS3NOS1NOS2ALDH1A1
SCHEMBL29492793 0.74 NOS3 (0.56) NOS3NOS1NOS2ALDH1A1
SCHEMBL5942438 0.74 ALDH1A1 (0.36) CYP3A4NOS3NOS1NOS2ALDH1A1
SCHEMBL19088190 0.74 ALDH1A1 (0.36) CYP3A4NOS3NOS1NOS2ALDH1A1
SCHEMBL5942363 0.74 PIK3CA (0.38) ALDH1A1
SCHEMBL31032811 0.74 PDE4A (0.38) HPGDALDH1A1F2GLAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920424-B1 NON-PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS WARNER LAMBERT CO (US) 2005-11-30 EP disclosed
US-6194437-B1 ANTIDEPRESSANTS; ANTICANCER AGENTS; GASTROINTESTINAL DISORDERS; COGNITION ACTIVATORS WARNER-LAMBERT COMPANY 2001-02-27 US disclosed
EP-0920424-A1 NON-PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1999-06-09 EP disclosed
WO-1998007718-A1 NON-PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-02-26 WO disclosed