SCHEMBL6185340

SCHEMBL6185340

CC(C)COc1ccccc1C=C[N+](=O)[O-]

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.59
MAPT P10636 7/20 0.59
LMNA P02545 4/20 0.59
NPSR1 Q6W5P4 4/20 0.59
HPGD P15428 3/20 0.59
RAB9A P51151 3/20 0.59
MAPK1 P28482 2/20 0.59
NPC1 O15118 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
S1PR4 O95977 1/20 0.59
ITGA4 P13612 1/20 0.59
S1PR1 P21453 1/20 0.59
TLR9 Q9NR96 1/20 0.59
TLR4 O00206 4/20 0.56
TLR2 O60603 4/20 0.56
PRMT1 Q99873 1/20 0.51
FBP1 P09467 6/20 0.50
NTSR1 P30989 2/20 0.50
ALOX12 P18054 1/20 0.50
CCR6 P51684 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185335 1.00 ALDH1A1 (0.59) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL27823272 0.83 ALDH1A1 (0.43) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL16499817 0.81 ALDH1A1 (0.60) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL16499818 0.81 ALDH1A1 (0.60) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL8002601 0.81 ALDH1A1 (0.64) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL3792354 0.80 TLR4 (0.60) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL3792351 0.80 TLR4 (0.60) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL793033 0.78 PRMT1 (0.73) ALDH1A1MAPTLMNANPSR1HPGD
SCHEMBL21915558 0.78 MEN1 (0.46) ALDH1A1MAPTLMNAHPGDSMN1; SMN2
SCHEMBL793032 0.78 PRMT1 (0.73) ALDH1A1MAPTLMNANPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-08-17 EP disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed