SCHEMBL6187038

SCHEMBL6187038

CC(=O)C(F)SC(c1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.50
SLC6A4 P31645 2/20 0.45
SLC6A3 Q01959 2/20 0.45
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
FFAR2 O15552 1/20 0.38
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
CNR2 P34972 1/20 0.36
POLB P06746 1/20 0.36
ADRB2 P07550 1/20 0.35
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 2/20 0.34
HSD17B10 Q99714 1/20 0.34
GABBR2 O75899 3/20 0.34
GABBR1 Q9UBS5 3/20 0.34
LMNA P02545 2/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6186523 0.77 BRD4 (0.45) BRD4SLC6A4SLC6A3FFAR2
SCHEMBL6188068 0.75 BRD4 (0.46) BRD4SLC6A4SLC6A3CES2CES1
SCHEMBL6192279 0.73 BRD4 (0.45) BRD4SLC6A4SLC6A3POLBCYP2C9
SCHEMBL10977277 0.73 SLC6A4 (0.52) BRD4SLC6A4SLC6A3HDAC4HDAC7
SCHEMBL6187976 0.73 ADRB2 (0.41) BRD4SLC6A4SLC6A3FFAR2POLB
SCHEMBL6186361 0.71 PPARG (0.43) BRD4SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL2788979 0.71 BRD4 (0.59) BRD4SLC6A4SLC6A3HDAC4HDAC7
SCHEMBL10882007 0.70 BRD4 (0.63) BRD4SLC6A4SLC6A3HDAC4HDAC7
SCHEMBL6185119 0.69 HPGD (0.46) BRD4CNR2POLBCYP2C19CYP3A4
SCHEMBL6075209 0.69 SLC6A3 (0.68) BRD4SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539685-A1 MCP-1 RECEPTOR ANTAGONISTS AND METHOD OF USE THEREOF Warner-Lambert Company LLC (US) 2005-06-15 EP disclosed
WO-2004014847-A1 MCP-1 RECEPTOR ANTAGONISTS AND METHOD OF USE THEREOF WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed