SCHEMBL6188736

SCHEMBL6188736

Cc1c(C(=O)c2c(Cl)cccc2Cl)[nH]c2ccc(NC(=O)C3CCCC3)cc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
NPSR1 Q6W5P4 1/20 0.49
JAK2 O60674 2/20 0.46
TYK2 P29597 2/20 0.46
STK17B O94768 1/20 0.46
STK17A Q9UEE5 1/20 0.46
ALDH1A1 P00352 2/20 0.45
ITK Q08881 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 2/20 0.44
JAK1 P23458 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185359 0.98 MAOA (0.48) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6185251 0.96 HPGD (0.47) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6185134 0.85 MAOA (0.54) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6186285 0.84 MAOA (0.49) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6189327 0.82 HPGD (0.46) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6187358 0.81 F2R (0.51) STK17BSTK17AALDH1A1KDM4EHPGD
SCHEMBL6188627 0.80 MAOB (0.47) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6186848 0.79 MAOB (0.49) MAOAMAOBNPSR1JAK2TYK2
SCHEMBL6186086 0.78 MAPT (0.39) MAOAMAOBJAK2ALDH1A1SMN1; SMN2
SCHEMBL6187129 0.78 GRM4 (0.51) MAOAMAOBNPSR1STK17BSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554271-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2005-07-20 EP disclosed
WO-2004035571-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2004-04-29 WO disclosed