SCHEMBL6188780

SCHEMBL6188780

COc1ccc(-c2[c]cccc2OC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
CLK4 Q9HAZ1 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HTT P42858 2/20 0.39
ESR2 Q92731 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
APP P05067 1/20 0.38
CA4 P22748 1/20 0.38
ABL1 P00519 2/20 0.38
ABCB1 P08183 2/20 0.38
BCR P11274 2/20 0.38
SYK P43405 2/20 0.38
AURKB Q96GD4 1/20 0.38
INCENP Q9NQS7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454339 0.85 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL8089505 0.85 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL215577 0.85 ADORA3 (0.43) CLK4ALDH1A1L3MBTL1SYKAURKB
SCHEMBL1274782 0.85 CA1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL2885322 0.82 CA1 (0.50) CA12CA1CA2CA7CA9
SCHEMBL1867724 0.81 ABL1 (0.50) CA12CA1CA2CA7CA9
SCHEMBL8089529 0.81 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL8089555 0.81 NPC1 (0.38) CA12CA1CA2CA7CA9
SCHEMBL10562502 0.81 CYP1A2 (0.43) CA12CA1CA2CA7CA9
SCHEMBL3411791 0.81 CYP1A1 (0.45) CA1CA2CA7CA9CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1601657-A1 PYRAZOLE MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2005-12-07 EP claimed
WO-2004080972-A1 PIRAZOLE MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-09-23 WO claimed
EP-0766664-A2 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1997-04-09 EP claimed
WO-1996009823-A9 HYPOGLYCEMIC AGENT FROM CRYPTOLEPIS 1996-05-23 WO claimed
WO-1996009823-A1 HYPOGLYCEMIC AGENT FROM CRYPTOLEPIS SHAMAN PHARMACEUTICALS, INC. (US) 1996-04-04 WO claimed
WO-1995035275-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1995-12-28 WO claimed
US-11635685-B2 Resist composition and patterning process SHIN-ETSU CHEMICAL CO., LTD. (JP) 2023-04-25 US disclosed
US-20210149300-A1 RESIST COMPOSITION AND PATTERNING PROCESS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2021-05-20 US disclosed
CN-110668950-A Chiral delta-nitroketene compound and asymmetric synthesis method and application thereof 浙江工业大学 2020-01-10 CN disclosed
CN-103827978-B Conductive composition, conductive member, method for producing same, touch panel, and solar cell FUJIFILM CORP. (JP) 2016-05-11 CN disclosed
EP-1289940-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001092213-A2 EXCITATORY AMINO ACID RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2001-12-06 WO disclosed
US-6124329-A AN ENZYME INHIBITOR FOR THE TREATMENT OR PROPHYLAXIS OF TISSUE BREAKDOWN, FOR EXAMPLE RHEUMATOID ARTHRITIS, OSTEOPOROSIS, PERIODONTITIS, GINGIVITIS, CORNEAL EPIDERMAL OR GASTRIC ULCERATION, AND TUMOR, MULTIPLE SCLEROSIS BRITISH BIOTECH PHARMACEUTICALS LTD. (GB) 2000-09-26 US disclosed
US-5962529-A OSTEOPOROSIS; RHEUMATIC DISORDERS; ORAL DISEASES; ANTIULCER AGENTS; ANTITUMOR AGENTS; ANTIINFLAMMATORY AGENTS; SKIN DISORDERS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1999-10-05 US disclosed
EP-0766664-A2 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1997-04-09 EP disclosed
WO-1996009823-A9 HYPOGLYCEMIC AGENT FROM CRYPTOLEPIS 1996-05-23 WO disclosed
WO-1995035275-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1995-12-28 WO disclosed
US-5461051-A Tetracyclic compounds having anti-allergic and anti-asthmatic activities and their use SANKYO COMPANY, LIMITED (JP) 1995-10-24 US disclosed