SCHEMBL6188801

SCHEMBL6188801

CCCC1(c2ccccc2)OC(=O)C(C(CC)c2cccc(O)c2)=C(O)C1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A1 O15245 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 2/20 0.34
OPRD1 P41143 2/20 0.34
ADRA2A P08913 2/20 0.34
ADRA2C P18825 2/20 0.34
DRD1 P21728 2/20 0.34
ADRA1A P35348 2/20 0.34
SLC6A3 Q01959 2/20 0.34
MLNR O43193 1/20 0.34
NR1I2 O75469 1/20 0.34
ABCB11 O95342 1/20 0.34
PGR P06401 1/20 0.34
CTSD P07339 1/20 0.34
CHRM2 P08172 1/20 0.34
PGA5 P0DJD9 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CTSE P14091 1/20 0.34
GABRA1 P14867 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6190123 0.91 CYP2C9 (0.37) OPRD1ADRA2AADRA2CDRD1ADRA1A
SCHEMBL6175249 0.77 MLNR (0.41) SLC22A1OPRM1OPRD1ADRA2AADRA2C
SCHEMBL6188998 0.76 OPRD1 (0.34) SLC22A1OPRM1OPRK1OPRD1SLC6A3
SCHEMBL7562120 0.76 ALDH1A1 (0.31) SLC22A1OPRM1OPRK1ALDH1A1HCAR3
SCHEMBL6188226 0.70 HTR2A (0.38) OPRD1ADRA2AADRA2CDRD1ADRA1A
SCHEMBL6173540 0.68 LDHA (0.40) OPRM1OPRK1OPRD1ADRA2AADRA2C
SCHEMBL25210900 0.68 CYP17A1 (0.55) SLC22A1OPRM1ADRA2AADRA2CDRD1
SCHEMBL27514771 0.68 SLC22A1 (0.57) SLC22A1OPRM1ADRA2AADRA2CDRD1
SCHEMBL6173274 0.67 OPRD1 (0.39) OPRM1OPRK1OPRD1ADRA2AADRA2C
SCHEMBL6948749 0.64 MLNR (0.49) OPRD1ADRA2AADRA2CDRD1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP claimed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed