SCHEMBL6189248

SCHEMBL6189248

CCCC1(CCCc2ccccc2)OC(=O)C(C(C=Cc2ccccc2)c2ccccc2)=C(O)C1=O

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
LMNA P02545 3/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4A O75164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HSD11B1 P28845 1/20 0.32
CNR2 P34972 1/20 0.32
EPHX2 P34913 2/20 0.31
SPHK1 Q9NYA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6189357 0.89 CNR2 (0.33) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6192154 0.87 CYP1A2 (0.34) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6191058 0.84 KDM4A (0.34) KDM4AHSD11B1EPHX2
SCHEMBL6191050 0.83 CYP1A2 (0.34) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6191220 0.82 KDM4A (0.33) CYP1A2CYP2C9CYP2C19KDM4AHSD11B1
SCHEMBL6188065 0.81 GAA (0.33) CYP3A4ALDH1A1LMNAKDM4EHSD17B10
SCHEMBL6174407 0.80 OPRD1 (0.43) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6174411 0.80 OPRD1 (0.43) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6188226 0.76 HTR2A (0.38) CYP2C9KDM4AHSD11B1EPHX2
SCHEMBL6174945 0.76 MLNR (0.48) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP claimed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed