SCHEMBL6192154

SCHEMBL6192154

CCCCC1(Cc2ccccc2)OC(=O)C(C(C=Cc2ccccc2)c2ccccc2)=C(O)C1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
TSHR P16473 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CNR2 P34972 1/20 0.32
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP8 P22894 2/20 0.32
MMP13 P45452 2/20 0.32
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HDAC3 O15379 2/20 0.31
EGFR P00533 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6189357 0.94 CNR2 (0.33) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6189248 0.87 CYP1A2 (0.34) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6186075 0.87 MMP2 (0.33) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6192554 0.82 MMP2 (0.36) CYP2C9KDM4EMMP2MMP9MMP8
SCHEMBL6191050 0.80 CYP1A2 (0.34) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6189549 0.80 MMP2 (0.34) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6174355 0.80 OPRD1 (0.36) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6174351 0.80 OPRD1 (0.36) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL6178709 0.75 MLNR (0.40) CYP1A2CNR2
SCHEMBL6178714 0.75 MLNR (0.40) CYP1A2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203770-B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases UPJOHN CO (US) 2005-03-09 EP claimed
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed