SCHEMBL6189800

SCHEMBL6189800

NC(=O)c1ccc(CNc2nc(CC(=O)N3CCN(Cc4ccc5c(c4)OCO5)CC3)nc(N3CCOCC3)n2)cc1-c1ccccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.43
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
PKM P14618 1/20 0.42
KDM4E B2RXH2 3/20 0.41
HTT P42858 3/20 0.41
LMNA P02545 5/20 0.40
TSHR P16473 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
USP2 O75604 2/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FAAH O00519 2/20 0.40
HDAC1 Q13547 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1058430 0.84 HDAC1 (0.62) KDM4ELMNAUSP2HDAC1
SCHEMBL13713693 0.78 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1PKMKDM4E
SCHEMBL1065171 0.76 KMT2A (0.52) ALDH1A1KMT2AMEN1PKMKDM4E
SCHEMBL3557879 0.74 HDAC1 (0.53) ALDH1A1KMT2AMEN1KDM4ELMNA
SCHEMBL10579147 0.65 FAAH (0.67) NR1H4ALDH1A1KMT2AMEN1PKM
SCHEMBL211529 0.65 HDAC1 (0.58) ALDH1A1KMT2APKMKDM4EHTT
SCHEMBL8346243 0.62 HDAC1 (0.54) HDAC1
SCHEMBL14503122 0.62 GALR2 (0.66) ALDH1A1KMT2AMEN1KDM4EHTT
SCHEMBL3142795 0.61 ALDH1A1 (0.72) ALDH1A1KMT2AMEN1KDM4EHTT
SCHEMBL7933991 0.61 ALDH1A1 (0.72) ALDH1A1KMT2AMEN1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1590340-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2005-11-02 EP disclosed
WO-2004069823-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2004-08-19 WO disclosed