SCHEMBL6195075

SCHEMBL6195075

CC(O)C(Oc1cccc2cccc(F)c12)N1CCNCC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.41
SLC6A4 P31645 14/20 0.41
KCNH2 Q12809 10/20 0.41
SLC6A3 Q01959 6/20 0.41
CYP2D6 P10635 3/20 0.40
HTR6 P50406 3/20 0.38
HRH4 Q9H3N8 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6260656 0.87 SLC6A2 (0.45) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL6192035 0.87 SLC6A2 (0.45) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL6193617 0.78 HTR6 (0.48) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL3634855 0.78 HTR6 (0.48) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL4605132 0.77 ADRB3 (0.46) SLC6A2SLC6A4KCNH2SLC6A3HTR6
SCHEMBL6185597 0.72 HRH3 (0.39) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL5901549 0.71 POLB (0.60)
SCHEMBL5995472 0.70 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3HTR2AHTR2C
SCHEMBL9330136 0.69 HTR2A (0.42) SLC6A2SLC6A4KCNH2CYP2D6HTR6
SCHEMBL16825719 0.68 ALDH1A1 (0.46) SLC6A2SLC6A4KCNH2SLC6A3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583751-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL IN THE TREATMENT OF CARDIOVASCULAR DISEASES CV THERAPEUTICS, INC. (US) 2005-10-12 EP disclosed
WO-2004069818-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL IN THE TREATMENT OF CARDIOVASCULAR DISEASES CV THERAPEUTICS INC. (US) 2004-08-19 WO disclosed