SCHEMBL619639

SCHEMBL619639

Cc1nc2ncccc2cc1C(=O)NCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
GALR3 O60755 1/20 0.56
NR2F2 P24468 1/20 0.56
SUCNR1 Q9BXA5 4/20 0.53
EGLN1 Q9GZT9 1/20 0.50
LMNA P02545 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
RAB9A P51151 1/20 0.47
HPGD P15428 3/20 0.46
NSD2 O96028 1/20 0.46
MMP13 P45452 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
KLKB1 P03952 1/20 0.46
KLK1 P06870 1/20 0.46
TACR3 P29371 1/20 0.46
EPHX2 P34913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10278163 0.93 EGLN1 (0.57) HTTSMN1; SMN2EGLN1LMNAKDM4E
SCHEMBL619854 0.92 HTT (0.52) HTTSMN1; SMN2GALR3NR2F2SUCNR1
SCHEMBL619835 0.91 HTT (0.49) HTTSMN1; SMN2GALR3NR2F2SUCNR1
SCHEMBL619376 0.91 LIPG (0.49) HTTSMN1; SMN2GALR3NR2F2SUCNR1
SCHEMBL616897 0.89 EGLN1 (0.60) HTTSMN1; SMN2SUCNR1EGLN1LMNA
SCHEMBL620070 0.89 HTT (0.54) HTTSMN1; SMN2GALR3NR2F2EGLN1
SCHEMBL619610 0.88 HTT (0.48) HTTSMN1; SMN2GALR3NR2F2SUCNR1
SCHEMBL619017 0.87 HTT (0.69) HTTSMN1; SMN2LMNARAB9AHPGD
SCHEMBL618734 0.87 EGLN1 (0.60) HTTSMN1; SMN2EGLN1LMNAALDH1A1
SCHEMBL616709 0.87 SMN1; SMN2 (0.54) HTTSMN1; SMN2EGLN1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 237 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-B1 NAPHTHYRIDINE DERIVATIVES HAVING BRONCHODILATING ACTIVITY RESPIRATORIUS AB (SE) 2013-07-24 EP claimed
US-8415333-B2 Bronchodilating diazaheteroaryls RESPIRATORIOUS AB (SE) 2013-04-09 US claimed
US-20120040942-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS RESPIRATORIUS AB (SE) 2012-02-16 US claimed
US-20090137567-A1 Methods for Treating Blood Disorders HEMAQUEST PHARMACEUTICALS, INC. (US) 2009-05-28 US claimed
EP-2023913-A2 METHODS FOR TREATING BLOOD DISORDERS Colorado State University Research Foundation (US) 2009-02-18 EP claimed
US-20080075692-A1 prophylaxis of blood disorder such as sickle cell anemia, beta -thalassemia, neutropenia or thrombocytopenia, comprising administering carboxylic acids, that stimulates production of fetal hemoglobin, hematopoiesis, erythropoiesis, myelopoiesis and neutrophil production COLORADO STATE UNIVERSITY RESEARCH FOUNDATION 2008-03-27 US claimed
WO-2007133653-A2 METHODS FOR TREATING BLOOD DISORDERS HEMAQUEST PHARMACEUTICALS, INC. (US) 2007-11-22 WO claimed
WO-2007006544-A2 CYCLIC ADENOSINE MONOPHOSPHATE COMPOUNDS FOR THE TREATMENT OF IMMUNE-RELATED DISORDERS VRIJE UNIVERSITEIT BRUSSEL (BE) 2007-01-18 WO claimed
EP-1546164-A4 (+)-TRANS-ISOMERS OF (1-PHOSPHONOMETHOXY-2-ALKYLCYCLOPROPYL) METHYL NUCLEOSIDE DERIVATIVES, PROCESS FOR THE PREPARATION OF STEREOISOMERS THEREOF, AND USE OF ANTIVIRAL AGENTS THEREOF LG LIFE SCIENCES LTD (KR) 2006-06-07 EP claimed
EP-1546164-A1 (+)-TRANS-ISOMERS OF (1-PHOSPHONOMETHOXY-2-ALKYLCYCLOPROPYL) METHYL NUCLEOSIDE DERIVATIVES, PROCESS FOR THE PREPARATION OF STEREOISOMERS THEREOF, AND USE OF ANTIVIRAL AGENTS THEREOF LG Life Sciences Ltd. (KR) 2005-06-29 EP claimed
WO-2004029064-A1 (+)-TRANS-ISOMERS OF (1-PHOSPHONOMETHOXY-2-ALKYLCYCLOPROPYL) METHYL NUCLEOSIDE DERIVATIVES, PROCESS FOR THE PREPARATION OF STEREOISOMERS THEREOF, AND USE OF ANTIVIRAL AGENTS THEREOF LG LIFE SCIENCES LTD. (KR) 2004-04-08 WO claimed
EP-1304325-A1 5-(M-CYANOBENZYLAMINO)PYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-04-23 EP claimed
US-6403633-B2 USEFUL ANTIANGIOGENIC, ANTIARTHRITIC, ANTIINFLAMMATORY, ANTIRESTENOTIC, ANTIINVASIVE, ANTIMETASTIC, ANTIOSTEOPOROTIC, ANTIRETINOPATHIC, CONTRACEPTIVE AND TUMORISTATIC TREATMENT AGENTS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-06-11 US claimed
US-5908930-A 5,10-dihydropyrimdo 4,5-b!quinolin-4(1H)-one tyrosine kinase inhibitors PFIZER INC. (US) 1999-06-01 US claimed
WO-1996028444-A1 5,10-DIHYDROPYRIMIDO[4,5-b]QUINOLIN-4(1H)-ONE TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1996-09-19 WO claimed
US-4650868-A 7-deazapurine derivatives useful as antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-03-17 US claimed
US-4138558-A Anthraquinone compounds NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1979-02-06 US claimed
US-12011490-B2 Dental photocurable composition excellent in operability and storage stability SHOFU INC. (JP) 2024-06-18 US disclosed
US-3962215-A PHOSPHORYLATION, ACYLATION, WATER, ACID CHLORIDE, ALCOHOL AMERICAN HOME PRODUCTS CORPORATION (US) 1976-06-08 US disclosed
US-3954732-A BACTERICIDAL PENICILLINS FUJISAWA PHARMACEUTICAL CO., LTD. (JA) 1976-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12011490-B2 Dental photocurable composition excellent in operability and storage stability H1-0, CCND1, CCNT1 HTT 932/4885SMN1; SMN2 1171/4885GALR3 2190/4885
US-20120040942-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS CHRM3, ADRB1, ADRB3 HTT 4219/4885SMN1; SMN2 4137/4885GALR3 246/4885
US-20090137567-A1 Methods for Treating Blood Disorders HBB, HBG1, HBG2 HTT 551/4885SMN1; SMN2 1168/4885GALR3 2878/4885
US-20080075692-A1 prophylaxis of blood disorder such as sickle cell anemia, beta -thalassemia, neutropenia or thrombocytopenia, comprising administering carboxylic acids, that stimulates production of fetal hemoglobin, hematopoiesis, erythropoiesis, myelopoiesis and neutrophil production HBG1, HBG2, HBB HTT 508/4885SMN1; SMN2 179/4885GALR3 3765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.