SCHEMBL6198213

SCHEMBL6198213

COC(=O)/C=C/c1c(-c2cccc(N3CCOCC3)c2)cc(Sc2cc(-c3cccc(N4CCOCC4)c3)c(/C=C/C(=O)OC)c(Cl)c2Cl)c(Cl)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.45
ALDH1A1 P00352 2/20 0.43
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 3/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
POLQ O75417 1/20 0.39
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6200061 0.89 KMO (0.43) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL6197595 0.81 ITGAL (0.46) POLBITGB2ICAM1ITGAL
SCHEMBL6201623 0.80 RAB9A (0.47) ALDH1A1KDM4ESMN1; SMN2MEN1POLB
SCHEMBL6195509 0.79 CCNC (0.36) ALDH1A1HTTKDM4ESMN1; SMN2MAPT
SCHEMBL6311336 0.79 POLB (0.44) POLBITGB2ICAM1ITGAL
SCHEMBL6318617 0.75 RAB9A (0.49) ALDH1A1KDM4ESMN1; SMN2POLBITGB2
SCHEMBL6318242 0.75 POLB (0.42) POLBITGB2ICAM1ITGALAKR1C3
SCHEMBL6317608 0.74 RAB9A (0.48) KDM4EPOLBITGB2ICAM1ITGAL
SCHEMBL6317511 0.74 LGMN (0.43) ALDH1A1KDM4ESMN1; SMN2MAPTMEN1
SCHEMBL6917194 0.73 RAB9A (0.52) SMN1; SMN2MEN1POLBKMT2AITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140814-B1 CELL ADHESION-INHIBITING ANTIINFLAMMATORY AND IMMUNE-SUPPRESSIVE COMPOUNDS ABBOTT LAB (US) 2005-05-25 EP disclosed