SCHEMBL6198397

SCHEMBL6198397

O=C(O)NC1CCN(c2ncnc3oc(-c4ccc(Cl)nc4)c(-c4ccc(F)cc4)c23)CC1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.50
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PAK1 Q13153 2/20 0.41
RPS6KB1 P23443 5/20 0.41
SSTR5 P35346 1/20 0.41
MAPT P10636 1/20 0.39
ADK P55263 1/20 0.38
MAP3K5 Q99683 1/20 0.38
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
STK4 Q13043 1/20 0.37
STK3 Q13188 1/20 0.37
LRRK2 Q5S007 1/20 0.37
CHRM4 P08173 1/20 0.37
MERTK Q12866 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848492 0.89 AURKA (0.44) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6846664 0.87 AURKA (0.55) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6200264 0.86 AURKA (0.64) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6203305 0.82 AURKA (0.49) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6199702 0.80 AURKA (0.78) AURKAALDH1A1HPGDTSHRHSD17B10
Hydrochloric Acid SCHEMBL6204384 0.79 AURKA (0.44) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6848519 0.78 CKS1B (0.43) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6198489 0.78 ALDH1A1 (0.47) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6203462 0.76 AURKA (0.42) AURKAALDH1A1HPGDTSHRHSD17B10
SCHEMBL6201006 0.76 AURKA (0.66) AURKAALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425283-B1 NOVEL 4-AMINOFUROPYRIMIDINES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2005-03-16 EP disclosed