SCHEMBL6199137

SCHEMBL6199137

O=c1ccn(CC(O)CO)c(C(O)c2ccccc2)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
TP53 P04637 2/20 0.40
CYP2D6 P10635 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
COMT P21964 2/20 0.33
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
ABCB1 P08183 1/20 0.33
MMP9 P14780 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
VEGFA P15692 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6195293 0.83 KDM4E (0.41) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6197640 0.82 KDM4E (0.46) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6198182 0.81 KMT2A (0.42) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL27481986 0.80 KMT2A (0.41) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6195550 0.79 HTT (0.47) HTTSMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL6197536 0.78 CYP2D6 (0.38) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6196471 0.76 KDM4E (0.41) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6200685 0.76 HTT (0.49) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6193890 0.75 LMNA (0.46) KDM4ETP53CYP2D6HTTSMN1; SMN2
SCHEMBL6949699 0.74 KDM4E (0.53) KDM4ETP53CYP2D6HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0768302-B1 Hydroxypyridinones NOVARTIS AG (CH) 2005-07-06 EP disclosed
US-5688815-A COMPOUNDS FOR REMOVAL OF EXCESS IRON IN MAMMALS CIBA GEIGY CORPORATION (US) 1997-11-18 US disclosed
EP-0768302-A2 Hydroxypyridinones Novartis AG (CH) 1997-04-16 EP disclosed