SCHEMBL6200321

SCHEMBL6200321

NC(C(=O)c1ccc(Cl)cc1)C(=O)c1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.54
CES1 P23141 3/20 0.54
TSHR P16473 2/20 0.52
ALOX15 P16050 1/20 0.52
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
LMNA P02545 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MAPT P10636 1/20 0.50
GSK3B P49841 2/20 0.46
SRD5A2 P31213 1/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27608931 0.90 KMT2A (0.47) CES2CES1TSHRALOX15CA1
SCHEMBL10964872 0.84 CES2 (0.52) CES2CES1TSHRALOX15CA1
Hydrochloric Acid SCHEMBL27977562 0.82 CES2 (0.50) CES2CES1TSHRALOX15CA1
SCHEMBL187689 0.82 CES2 (0.50) CES2CES1TSHRALOX15CA1
SCHEMBL6205327 0.81 MDM2 (0.45) CES2CES1ALOX15ALDH1A1RAB9A
Hydrochloric Acid SCHEMBL10809276 0.80 CES2 (0.48) CES2CES1TSHRALOX15CA1
SCHEMBL27608836 0.80 CES2 (0.48) CES2CES1TSHRALOX15CA1
SCHEMBL20263132 0.80 SMN1; SMN2 (0.50) CES2CES1TSHRCA1CA2
SCHEMBL655925 0.79 LMNA (0.48) CES2CES1TSHRALOX15CA1
Hydrochloric Acid SCHEMBL9150527 0.79 CES2 (0.46) CES2CES1TSHRALOX15CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed