SCHEMBL6205327

SCHEMBL6205327

NC(C(=O)c1ccc(Cl)cc1)C(=O)c1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 9/20 0.45
CES2 O00748 3/20 0.45
CES1 P23141 3/20 0.45
MGLL Q99685 1/20 0.45
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
NR4A1 P22736 1/20 0.42
RAB9A P51151 1/20 0.41
KCNMA1 Q12791 1/20 0.40
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6200321 0.81 CES2 (0.54) CES2CES1ALDH1A1ALOX15SMN1; SMN2
SCHEMBL29779621 0.76 NR4A1 (0.65) CES2CES1MGLLALDH1A1ALOX15
SCHEMBL1129231 0.76 NR4A1 (0.65) CES2CES1MGLLALDH1A1ALOX15
SCHEMBL9421742 0.75 NR4A1 (0.62) CES2CES1MGLLALDH1A1ALOX15
SCHEMBL27608931 0.73 KMT2A (0.47) CES2CES1MGLLALDH1A1ALOX15
SCHEMBL6203257 0.72 RAB9A (0.52) ALDH1A1SMN1; SMN2RAB9A
SCHEMBL9861760 0.70 ALDH1A1 (0.59) CES2CES1ALDH1A1ALOX15SMN1; SMN2
SCHEMBL20659167 0.69 MGLL (0.44) CES2CES1MGLLALDH1A1ALOX15
SCHEMBL9450434 0.69 TDP1 (0.56) MDM2CES2CES1ALDH1A1ALOX15
SCHEMBL11184715 0.69 KMT2A (0.61) CES2CES1ALDH1A1ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed