SCHEMBL6201328

SCHEMBL6201328

NCCc1cccc(Oc2cncnc2)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.56
ACHE P22303 3/20 0.46
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43
CHRNA7 P36544 1/20 0.43
MAOB P27338 1/20 0.41
HTR2C P28335 1/20 0.39
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201445 0.86 LMNA (0.64) TAAR1ACHELMNATDP1DRD2
SCHEMBL6204785 0.82 TAAR1 (0.57) TAAR1ACHEDRD2DRD1CHRNA7
SCHEMBL415399 0.81 TAAR1 (0.65) TAAR1ACHEDRD2DRD1MAOB
Hydrochloric Acid SCHEMBL5356526 0.80 TAAR1 (0.62) TAAR1ACHEMAOBHTR2CHTR6
SCHEMBL29102430 0.77 TAAR1 (0.86) TAAR1MAOB
SCHEMBL30631696 0.77 TAAR1 (0.86) TAAR1MAOB
SCHEMBL6203524 0.76 TAAR1 (0.50) TAAR1ACHECHRNA7MAOB
SCHEMBL6203586 0.76 TAAR1 (0.54) TAAR1ACHELMNATDP1MAOB
SCHEMBL6199971 0.75 TAAR1 (0.62) TAAR1ACHEDRD2DRD1MAOB
SCHEMBL5947233 0.73 CYP1A2 (0.51) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581498-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS Bristol-Myers Squibb Company (US) 2005-10-05 EP disclosed
WO-2004047739-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-10 WO disclosed