SCHEMBL6202500

SCHEMBL6202500

O=C(Cc1ccccc1F)c1ccc(Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.59
MAPT P10636 2/20 0.59
TDP1 Q9NUW8 1/20 0.56
RAB9A P51151 6/20 0.51
NPC1 O15118 5/20 0.51
CNR1 P21554 1/20 0.51
ALDH1A1 P00352 3/20 0.49
MAPK1 P28482 1/20 0.49
GSK3B P49841 2/20 0.48
PPARG P37231 1/20 0.48
PPARA Q07869 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
HTT P42858 1/20 0.47
HSD11B1 P28845 1/20 0.45
RECQL P46063 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29533518 0.85 MAPK1 (0.54) L3MBTL1MAPTTDP1RAB9AALDH1A1
SCHEMBL70282 0.85 MAPK1 (0.54) L3MBTL1MAPTTDP1RAB9AALDH1A1
SCHEMBL7265238 0.83 ALDH1A1 (0.49) L3MBTL1MAPTTDP1RAB9AALDH1A1
SCHEMBL28061321 0.83 ALDH1A1 (0.49) MAPTRAB9ANPC1ALDH1A1MAPK1
SCHEMBL2085224 0.82 L3MBTL1 (0.62) L3MBTL1MAPTRAB9ANPC1CNR1
SCHEMBL1025697 0.81 MAPT (0.56) L3MBTL1MAPTRAB9ANPC1CNR1
SCHEMBL17459291 0.80 KMT2A (0.53) L3MBTL1MAPTTDP1RAB9ACNR1
SCHEMBL3282677 0.79 ALDH1A1 (0.53) L3MBTL1RAB9AALDH1A1MAPK1GSK3B
SCHEMBL2571844 0.78 L3MBTL1 (0.62) L3MBTL1MAPTRAB9ANPC1ALDH1A1
SCHEMBL10046960 0.77 ALDH1A1 (0.51) L3MBTL1MAPTTDP1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
US-5532374-A Method of preparation of bis-quinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1996-07-02 US disclosed