SCHEMBL6202658

SCHEMBL6202658

CC(C)N(CCO)c1nc(Nc2ccc(O)c(C(=O)O)c2)c2c(n1)N(C(C)C)NN2C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.44
CTNNB1 P35222 1/20 0.36
GAA P10253 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
XDH P47989 1/20 0.35
USP2 O75604 1/20 0.35
PKM P14618 1/20 0.35
CDK5 Q00535 3/20 0.35
CDK5R1 Q15078 3/20 0.35
DDX3X O00571 1/20 0.35
CCNE2 O96020 4/20 0.33
CCNE1 P24864 4/20 0.33
CDK2 P24941 4/20 0.33
ALDH1A1 P00352 2/20 0.33
AMY1A P0DUB6 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CCNB2 O95067 1/20 0.33
NTRK1 P04629 1/20 0.33
INSR P06213 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203872 0.91 CDK1 (0.44) CDK1GAAMEN1KMT2ACDK5
SCHEMBL6205009 0.89 CDK5 (0.44) CDK1MEN1KMT2ACDK5CDK5R1
SCHEMBL6203387 0.82 CCNE2 (0.38) CDK1CDK5CDK5R1CCNE2CCNE1
SCHEMBL6205532 0.81 CDK5 (0.35) CDK1CDK5CDK5R1CCNE2CCNE1
SCHEMBL6202790 0.81 CDK5 (0.35) CDK1CDK5CDK5R1CCNE2CCNE1
SCHEMBL6206176 0.80 CDK5 (0.49) CDK1MEN1KMT2ACDK5CDK5R1
SCHEMBL3444586 0.80 CDK1 (0.63) CDK1GAAMEN1KMT2AXDH
SCHEMBL3445408 0.78 CDK1 (0.44) CDK1CTNNB1GAAMEN1KMT2A
SCHEMBL3445200 0.78 CDK1 (0.49) CDK1CDK5CDK5R1CCNE2CCNE1
SCHEMBL6201043 0.77 CDK1 (0.40) CDK1CTNNB1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed