SCHEMBL6202944

SCHEMBL6202944

NCCOc1cccc(OCCOc2nccnc2N2CCNCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.39
EPHX2 P34913 1/20 0.38
HTR6 P50406 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
ADRB1 P08588 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
PIM1 P11309 1/20 0.37
PIM3 Q86V86 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4308724 0.91 EPHX2 (0.40) HTR2CEPHX2HTR6HTR1ASLC6A2
SCHEMBL4311413 0.88 TSHR (0.40) HTR2CEPHX2ADRB1CYP3A4
SCHEMBL4315672 0.88 ADRB1 (0.52) HTR2CHTR6HTR1AADRB1CHRNB2
SCHEMBL4313451 0.88 KDM4E (0.39) HTR2CEPHX2HTR6HTR1ASLC6A2
SCHEMBL2640084 0.88 CHRNB2 (0.49) HTR2CHTR6ADRB1CHRNB2CHRNA4
SCHEMBL4320133 0.87 HTR2C (0.42) HTR2CHTR6ADRB1CHRNB2CHRNA4
SCHEMBL4325739 0.86 HTR2C (0.38) HTR2CEPHX2HTR6HTR1ASLC6A2
SCHEMBL4318628 0.86 HTT (0.42) KDM4EALDH1A1
SCHEMBL4316517 0.86 HTR1A (0.53) HTR2CEPHX2HTR6HTR1ASLC6A2
SCHEMBL4308710 0.86 CHRNB4 (0.40) HTR2CHTR1ASLC6A2SLC6A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178973-B1 PYRAZINYL-PIPERAZINE- COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2005-12-21 EP disclosed