SCHEMBL6203203

SCHEMBL6203203

CCCN(CO)c1nc(Nc2ccc(C(=O)O)c(Cl)c2)c2nn[nH]c2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
CDK1 P06493 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CCNB2 O95067 1/20 0.40
CCNE2 O96020 1/20 0.40
ALDH1A1 P00352 1/20 0.40
NTRK1 P04629 1/20 0.40
INSR P06213 1/20 0.40
CCNB1 P14635 1/20 0.40
PRKACA P17612 1/20 0.40
CCNA2 P20248 1/20 0.40
PRKACG P22612 1/20 0.40
PRKACB P22694 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
MAPK3 P27361 1/20 0.40
CCNA1 P78396 1/20 0.40
NTRK2 Q16620 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203207 0.86 KDM4E (0.36) CDK5CDK5R1CDK1KDM4ECCNB2
SCHEMBL6205210 0.86 HTR2A (0.35) CDK5CDK5R1HTR2AHTR2CATM
SCHEMBL6204174 0.84 HTR2A (0.35) CDK5CDK5R1HTR2AHTR2CATM
SCHEMBL6202086 0.83 HTR2C (0.48) CDK5CDK5R1KDM4ECCNE2ALDH1A1
SCHEMBL6205643 0.82 CDK5 (0.45) CDK5CDK5R1CDK1KDM4ECCNB2
SCHEMBL6203247 0.81 CCNE2 (0.43) CCNE2CCNE1CDK2HTR2AHTR2C
SCHEMBL6204146 0.80 CCNE2 (0.45) CDK1KDM4ECCNE2CCNE1CDK2
SCHEMBL6203210 0.77 CCNE2 (0.42) CDK5CDK5R1CDK1KDM4ECCNB2
SCHEMBL3446235 0.76 CDK5 (0.51) CDK5CDK5R1CDK1KDM4ECCNB2
SCHEMBL3446217 0.74 CDK5 (0.66) CDK5CDK5R1CDK1KDM4ECCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed