SCHEMBL6205643

SCHEMBL6205643

CCCN(CO)c1nc(Nc2cccc(Cl)c2)c2nn[nH]c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 4/20 0.45
CDK5R1 Q15078 4/20 0.45
ATM Q13315 1/20 0.45
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CDK1 P06493 5/20 0.39
CFTR P13569 2/20 0.38
HTR2C P28335 3/20 0.37
HTR2A P28223 2/20 0.37
KDM4E B2RXH2 3/20 0.37
NPC1 O15118 2/20 0.37
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
CCNB1 P14635 3/20 0.36
GRM4 Q14833 1/20 0.36
EIF2AK2 P19525 1/20 0.36
GSK3B P49841 1/20 0.36
MERTK Q12866 1/20 0.36
FADS1 O60427 3/20 0.36
CCNB2 O95067 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202086 0.88 HTR2C (0.48) CDK5CDK5R1ATMMEN1KMT2A
SCHEMBL6203247 0.87 CCNE2 (0.43) MEN1KMT2ACFTRHTR2CHTR2A
SCHEMBL6205647 0.85 CDK5 (0.41) CDK5CDK5R1ATMMEN1KMT2A
SCHEMBL6204174 0.84 HTR2A (0.35) CDK5CDK5R1ATMMEN1KMT2A
SCHEMBL6205210 0.84 HTR2A (0.35) CDK5CDK5R1ATMMEN1KMT2A
SCHEMBL6203203 0.82 CDK5 (0.40) CDK5CDK5R1ATMCDK1HTR2C
SCHEMBL6204146 0.81 CCNE2 (0.45) CDK1HTR2CHTR2AKDM4ENPC1
SCHEMBL3444401 0.75 MEN1 (0.48) MEN1KMT2ACDK1KDM4EMAPT
SCHEMBL6202754 0.75 CDK5 (0.43) CDK5CDK5R1MEN1KMT2ACDK1
SCHEMBL6204714 0.74 SLC29A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed