SCHEMBL6202086

SCHEMBL6202086

CCCN(CO)c1nc(Nc2ccc(Cl)cc2)c2nn[nH]c2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.48
HTR2A P28223 3/20 0.48
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CCNE2 O96020 3/20 0.34
CCNE1 P24864 3/20 0.34
CDK2 P24941 3/20 0.34
LMNA P02545 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CRHR1 P34998 2/20 0.33
CNR1 P21554 1/20 0.33
POLB P06746 1/20 0.33
RXRA P19793 1/20 0.33
NR4A2 P43354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204146 0.89 CCNE2 (0.45) HTR2CHTR2AMAPTNPSR1CCNE2
SCHEMBL6203247 0.89 CCNE2 (0.43) HTR2CHTR2AMEN1KMT2ANPSR1
SCHEMBL6205643 0.88 CDK5 (0.45) HTR2CHTR2AMEN1KMT2AMAPT
SCHEMBL6205210 0.86 HTR2A (0.35) HTR2CHTR2AMEN1KMT2ALMNA
SCHEMBL6204174 0.86 HTR2A (0.35) HTR2CHTR2AMEN1KMT2ALMNA
SCHEMBL6202094 0.84 HTR2C (0.47) HTR2CHTR2AMEN1KMT2AMAPT
SCHEMBL6203203 0.83 CDK5 (0.40) HTR2CHTR2ACCNE2CCNE1CDK2
SCHEMBL6202754 0.76 CDK5 (0.43) MEN1KMT2ASMN1; SMN2CCNE2CCNE1
SCHEMBL6204126 0.76 SLC29A1 (0.32)
SCHEMBL6204714 0.74 SLC29A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed