SCHEMBL6203415

SCHEMBL6203415

CCOC(OCC)c1ccnc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
RECQL P46063 1/20 0.39
LOX P28300 1/20 0.39
LOXL3 P58215 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
ACHE P22303 6/20 0.35
PTGS2 P35354 6/20 0.35
BCHE P06276 5/20 0.35
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
TRPA1 O75762 1/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
PFKFB3 Q16875 1/20 0.32
SMARCA2 P51531 1/20 0.31
SMARCA4 P51532 1/20 0.31
SLC6A3 Q01959 1/20 0.31
AAK1 Q2M2I8 2/20 0.31
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4651277 0.79 RECQL (0.38) RECQLLOXLOXL3LOXL2TRPA1
SCHEMBL16011482 0.79 NPC1 (0.40) NPC1RAB9AACHEPTGS2BCHE
SCHEMBL6206078 0.76 NPC1 (0.39) NPC1RAB9AACHEPTGS2BCHE
SCHEMBL20096333 0.76 RECQL (0.42) RECQLLOXLOXL3LOXL2AKR1C3
SCHEMBL23376898 0.74 RECQL (0.41) NPC1RAB9ARECQLLOXLOXL3
SCHEMBL12695310 0.74 RECQL (0.41) NPC1RAB9ARECQLLOXLOXL3
SCHEMBL18699316 0.74 RECQL (0.41) NPC1RAB9ARECQLLOXLOXL3
SCHEMBL27146027 0.74 RECQL (0.38) RECQLLOXLOXL3LOXL2AKR1C3
SCHEMBL2370569 0.73 MMP8 (0.41) RECQLAKR1C3AKR1C2SMARCA2SMARCA4
SCHEMBL6204290 0.73 NPC1 (0.37) NPC1RAB9AACHEPTGS2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107820494-A Nuclear receptor modulators 艾伯维公司 2018-03-20 CN disclosed
EP-1551841-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SmithKline Beecham Corporation (US) 2005-07-13 EP disclosed
WO-2004009602-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-01-29 WO disclosed
EP-0282077-B1 Pyridyloxy derivatives FUJIREBIO KK (JP) 1993-11-10 EP disclosed
US-4977267-A ANTISECRETORY AGENT FUJIREBIO KABUSHIKI KAISHA (JP) 1990-12-11 US disclosed
US-4912101-A Containing a secondary amide, suflur group and a furan ring FUJIREBIO KABUSHIKI KAISHA (JP) 1990-03-27 US disclosed
EP-0282077-A2 Pyridyloxy derivatives FUJIREBIO KABUSHIKI KAISHA (JP) 1988-09-14 EP disclosed