SCHEMBL6203942

SCHEMBL6203942

CC(C)(C)OC(=O)NCCc1cccc(Oc2ccncc2)c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 3/20 0.47
NQO2 P16083 1/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.44
KDM4E B2RXH2 1/20 0.44
NAMPT P43490 1/20 0.42
GLI1 P08151 1/20 0.42
GLI2 P10070 1/20 0.42
IDO1 P14902 1/20 0.41
CA2 P00918 1/20 0.41
AKR1C3 P42330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354570 0.90 FDFT1 (0.57) FDFT1NQO2NAMPTGLI1GLI2
SCHEMBL21090366 0.87 FDFT1 (0.47) FDFT1NQO2POLBKDM4ENAMPT
SCHEMBL6202190 0.86 PLAAT3 (0.48) FDFT1NQO2POLBKDM4ENAMPT
SCHEMBL6202759 0.84 PLAAT3 (0.52) NQO2POLBCYP3A4KDM4E
SCHEMBL6204512 0.83 FDFT1 (0.43) FDFT1NQO2POLBKDM4ENAMPT
SCHEMBL21090363 0.83 CYP4F2 (0.49) FDFT1NQO2CA2AKR1C3
SCHEMBL6204579 0.83 MTNR1A (0.58) POLBCA2
SCHEMBL2024124 0.81 CYP17A1 (0.53) NQO2CYP3A4KDM4ENAMPTCA2
SCHEMBL9889553 0.80 EPHX2 (0.52) NQO2POLBNAMPTCA2
SCHEMBL29828661 0.80 MTNR1A (0.48) NQO2POLBNAMPTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581498-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS Bristol-Myers Squibb Company (US) 2005-10-05 EP disclosed
WO-2004047739-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-10 WO disclosed