SCHEMBL6204512

SCHEMBL6204512

CC(C)(C)OC(=O)NCCc1cccc(Oc2ccccn2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FDFT1 P37268 2/20 0.43
POLB P06746 1/20 0.43
NQO2 P16083 1/20 0.43
NAMPT P43490 1/20 0.42
KDM4E B2RXH2 1/20 0.42
IDO1 P14902 1/20 0.42
MGLL Q99685 1/20 0.41
AKT1 P31749 1/20 0.41
GLS O94925 1/20 0.41
PLAAT3 P53816 1/20 0.40
PLAAT5 Q96KN8 1/20 0.40
PLAAT2 Q9NWW9 1/20 0.40
PLAAT4 Q9UL19 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202190 0.88 PLAAT3 (0.48) FDFT1POLBNQO2NAMPTKDM4E
SCHEMBL6202759 0.87 PLAAT3 (0.52) POLBNQO2KDM4EPLAAT3PLAAT5
SCHEMBL5354570 0.85 FDFT1 (0.57) FDFT1NQO2NAMPTIDO1PLAAT3
SCHEMBL6203942 0.83 FDFT1 (0.47) FDFT1POLBNQO2NAMPTKDM4E
SCHEMBL21090366 0.82 FDFT1 (0.47) FDFT1POLBNQO2NAMPTKDM4E
SCHEMBL31506266 0.81 CYP2D6 (0.58) NQO2KDM4EIDO1
SCHEMBL67569 0.81 CYP2D6 (0.58) NQO2KDM4EIDO1
SCHEMBL6204579 0.80 MTNR1A (0.58) POLB
SCHEMBL21090363 0.78 CYP4F2 (0.49) FDFT1NQO2
SCHEMBL3026698 0.77 CYP2D6 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581498-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS Bristol-Myers Squibb Company (US) 2005-10-05 EP disclosed
WO-2004047739-A2 PYRIDINYL, PYRIMIDINYL AND PYRAZINYL AMIDES AS POTASSIUM CHANNEL OPENERS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-10 WO disclosed