SCHEMBL6203832

SCHEMBL6203832

CC(=O)c1cccc(CNc2nc(C(C)C)nc3c2nnn3C(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
SRC P12931 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.36
CDK1 P06493 7/20 0.36
CCNB2 O95067 4/20 0.36
CCNB1 P14635 4/20 0.36
CCNB3 Q8WWL7 4/20 0.36
HDAC6 Q9UBN7 1/20 0.35
CDK2 P24941 2/20 0.35
PDE8B O95263 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226169 0.83 KMT2A (0.56) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL6202355 0.80 ALDH1A1 (0.46) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL6203983 0.76 KMT2A (0.42) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL3445315 0.73 CDK1 (0.49) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6201910 0.73 ALDH1A1 (0.49) KMT2AALDH1A1LMNASMN1; SMN2CDK1
SCHEMBL6203399 0.72 KMT2A (0.42) KMT2AALDH1A1LMNASMN1; SMN2CDK2
SCHEMBL3445310 0.72 CDK2 (0.49) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL3445903 0.71 CDK2 (0.43) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL3445486 0.71 CYP3A4 (0.54) KMT2AALDH1A1SMN1; SMN2CDK1KDM4E
SCHEMBL3444705 0.70 CDK1 (0.64) KMT2ACDK1CCNB2CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed