SCHEMBL6204310

SCHEMBL6204310

Cc1cccc(NS(=O)(=O)CC(=O)c2ccccc2)c1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
RAB9A P51151 2/20 0.49
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
AKR1B10 O60218 1/20 0.46
TRPA1 O75762 1/20 0.46
ABCB11 O95342 1/20 0.46
DHFR P00374 1/20 0.46
LMNA P02545 1/20 0.46
MPO P05164 1/20 0.46
CHRM1 P11229 1/20 0.46
AKR1B1 P15121 1/20 0.46
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
AKR1C3 P42330 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204418 0.78 KMT2A (0.50) RAB9AMEN1KMT2ATDP1CYP3A4
SCHEMBL27608803 0.76 RAB9A (0.48) KEAP1NFE2L2RAB9AMEN1KMT2A
SCHEMBL6202161 0.75 HPGD (0.56) KEAP1RAB9AMEN1KMT2ATDP1
SCHEMBL6205498 0.75 RECQL (0.60) RAB9AMEN1KMT2ATDP1LMNA
SCHEMBL6203277 0.74 NPC1 (0.59) RAB9AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL6202058 0.74 RECQL (0.49) RAB9AMEN1KMT2ATDP1LMNA
SCHEMBL11672581 0.71 KEAP1 (0.69) KEAP1NFE2L2RAB9AMEN1KMT2A
SCHEMBL11769542 0.70 POLB (0.77) RAB9AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL30288146 0.70 POLB (0.77) RAB9AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL5320792 0.70 RAB9A (0.65) RAB9AMEN1KMT2ATDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US claimed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP claimed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO claimed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed