SCHEMBL6204399

SCHEMBL6204399

Cc1ccc(S(=O)(=O)N(CC(=O)c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.67
NFE2L2 Q16236 2/20 0.67
RECQL P46063 1/20 0.56
KMT2A Q03164 3/20 0.55
MAPT P10636 1/20 0.55
PPARG P37231 1/20 0.54
PTGES O14684 3/20 0.54
ALOX5 P09917 2/20 0.54
CA12 O43570 1/20 0.53
CA9 Q16790 1/20 0.53
CNR1 P21554 1/20 0.52
CNR2 P34972 1/20 0.52
MEN1 O00255 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ESR1 P03372 1/20 0.51
HCRTR2 O43614 1/20 0.51
OXTR P30559 1/20 0.51
AVPR1A P37288 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL699184 0.87 KEAP1 (0.88) KEAP1NFE2L2KMT2APPARGCA12
SCHEMBL28561073 0.84 KEAP1 (0.61) KEAP1NFE2L2KMT2AMAPTPPARG
SCHEMBL6204172 0.84 ESR1 (0.55) KEAP1NFE2L2RECQLKMT2AMAPT
SCHEMBL14145796 0.84 RECQL (0.60) KEAP1NFE2L2RECQLKMT2APTGES
SCHEMBL11603483 0.82 RECQL (0.59) KEAP1NFE2L2RECQLKMT2ACA12
SCHEMBL5568657 0.82 NR1I2 (0.65) KEAP1NFE2L2KMT2APPARGMEN1
SCHEMBL28575718 0.82 KEAP1 (0.61) KEAP1NFE2L2KMT2AMAPTPPARG
SCHEMBL14502622 0.79 KEAP1 (0.66) KEAP1NFE2L2KMT2AMAPTPPARG
SCHEMBL28564469 0.79 LMNA (0.54) KEAP1NFE2L2KMT2AMAPTPPARG
SCHEMBL5604160 0.79 ESR1 (0.73) KEAP1NFE2L2KMT2AMAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed